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Home | About and More Information | Transporter Data Index |
No substrate information.
Transporter | Synonyms | Inhibitor | IC50 (μM) | Ki (μM) | Substrate used | Cell System | Reference |
---|---|---|---|---|---|---|---|
SLC22A2 | OCT2 | Vecuronium bromide | 3.5 | 4-(4-dimethylamino)styryl-N-methylpyridinium (ASP+) | HEK293-OCT2 | Wittwer, 2013 | |
SLC47A1 | MATE1 | Vecuronium bromide | 1.9 | 4-(4-dimethylamino)styryl-N-methylpyridinium (ASP+) | HEK293-MATE1 | Wittwer, 2013 | |
SLC47A2 | MATE2K | Vecuronium bromide | 25.2 | 4-(4-dimethylamino)styryl-N-methylpyridinium (ASP+) | HEK293-MATE2K | Wittwer, 2013 | |
ABCC2 | MRP2, cMOAT | Vecuronium bromide | >133 | Estradiol-17beta-glucuronide | Sf9 cell membrane vesicles | Morgan, 2013 | |
ABCC3 | MRP3 | Vecuronium bromide | >133 | Estradiol-17beta-glucuronide | Sf9 cell membrane vesicles | Morgan, 2013 | |
ABCC4 | MRP4 | Vecuronium bromide | >133 | Estradiol-17beta-glucuronide | Sf9 cell membrane vesicles | Morgan, 2013 | |
ABCB11 | BSEP | Vecuronium bromide | >133 | Taurocholate | Sf9 cell membrane vesicles | Morgan, 2013 |
No drug-drug interaction information.
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