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Trequinsin

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

No substrate information.


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In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
ABCC5 MRP5 Trequinsin 580 5-fluorodeoxyuridine monophosphate MRP5-expressing HEK293 vesicles Pratt, 2005
ABCC4 MRP4 Trequinsin 10 9-(2-phosphonomethoxyethyl)adenine (PMEA) MRP4-expressing HEK293 vesicles Reid, 2003
ABCC5 MRP5 Trequinsin 30 9-(2-phosphonomethoxyethyl)adenine (PMEA) MRP4-expressing HEK293 vesicles Reid, 2003
ABCC5 MRP5 Trequinsin 218 Carboxydichlorofluorescein MRP5-expressing HEK293 vesicles Pratt, 2006
ABCC5 MRP5 Trequinsin 0.24 Cyclic GMP MRP5-expressing V79 vesicles Jedlitschky, 2000

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Clinical Drug-Drug Interactions

No drug-drug interaction information.


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