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Home | About and More Information | Transporter Data Index |
No substrate information.
Transporter | Synonyms | Inhibitor | IC50 (μM) | Ki (μM) | Substrate used | Cell System | Reference |
---|---|---|---|---|---|---|---|
SLCO2B1 | OATP2B1, OATP-B | Tipranavir | 0.2 | Dibromofluorescein | HEK293-OATP2B1 | Unger, 2020 | |
SLCO1B1 | OATP1B1, OATP-C, OATP2, LST-1 | Tipranavir | 1.1 | Estradiol-17beta-glucuronide | HEK-OATP1B1 | Yoshida, 2012 | |
SLCO2B1 | OATP2B1, OATP-B | Tipranavir | 0.88 | Estrone sulfate | MDCK II-OATP2B1 | Kis, 2010 |
No drug-drug interaction information.
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