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Tetramethrin

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

No substrate information.


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In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
SLC22A1 OCT1 Tetramethrin 4.9 4',6'-diamidino-2-phenylindole HEK293 cells Chedik, 2017
ABCC2 MRP2, cMOAT Tetramethrin 65.5 Carboxy-2',7'-dichlorofluorescein diacetate HuH-7 cells Chedik, 2017
SLCO1B1 OATP1B1, OATP-C, OATP2, LST-1 Tetramethrin 5.7 Estrone sulfate CHO cells Chedik, 2017
SLC22A8 OAT3 Tetramethrin 77.6 Fluorescein HEK293 cells Chedik, 2017
ABCG2 BCRP, MXR Tetramethrin 72.5 Hoechst 33342 HEK293 cells Chedik, 2017
SLC22A2 OCT2 Tetramethrin 11.2 Rhodamine 123 HEK293 cells Chedik, 2017
SLC47A1 MATE1 Tetramethrin 47.5 Tetraethylammonium HEK293 cells Chedik, 2017

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Clinical Drug-Drug Interactions

No drug-drug interaction information.


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