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Sulpiride

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Km (μM) Cell System Reference
SLC22A2 OCT2 187.2 HEK293-OCT2 Dos, 2014
SLC22A1 OCT1 259.7 HEK293-OCT1 Dos, 2014
SLC22A1 OCT1 2.6 HEK293-OCT1 Takano, 2017
SLC22A2 OCT2 68 HEK293-OCT2 Takano, 2017
SLC47A1 MATE1 14.5 MDCK-MATE1 Li, 2017
SLC47A2 MATE2K 25.5 MDCK-MATE1 Li, 2017
SLC22A5 OCTN2 235 MDCK-hOCTN2 Li, 2017
SLC22A4 OCTN1 250 MDCK-hOCTN1 Li, 2017
SLC22A2 OCT2 390 MDCK-OCT2 Li, 2017

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In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
SLC22A1 OCT1 Sulpiride 182 Tetraethylammonium HEK293-OCT1 Takano, 2017

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Clinical Drug-Drug Interactions

No drug-drug interaction information.


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