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Rilpivirine

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

No substrate information.


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In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
SLCO1B1 OATP1B1, OATP-C, OATP2, LST-1 Rilpivirine 4.1 8-fluorescein-cAMP HEK-OATP1B1 Weiss, 2013
SLCO1B3 OATP1B3, OATP8 Rilpivirine 6.1 8-fluorescein-cAMP HEK293-OATP1B3 Weiss, 2013
ABCG2 BCRP, MXR Rilpivirine 1.5 Pheophorbide A polarized MDCKII-BCRP Weiss, 2013

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Clinical Drug-Drug Interactions

No drug-drug interaction information.


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