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Rhodamine 123

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Km (μM) Cell System Reference
ABCB1 MDR1, P-gp 21 ATPase assay of Sf9-MDR1 liposomes Kimura, 2007
SLC22A1 OCT1 0.54 HEK293-OCT1 Jouan, 2014

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In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
SLC22A1 OCT1 Rhodamine 123 0.37 Tetraethylammonium HEK293-OCT1 Jouan, 2014
ABCB1 MDR1, P-gp Rhodamine 123 0.5 Verapamil Caco-2 cells Doppenshmitt, 1998

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Clinical Drug-Drug Interactions

No drug-drug interaction information.


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