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Rapamycin

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

No substrate information.


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In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
SLCO1B3 OATP1B3, OATP8 Rapamycin 0.4 FMTX CHO-OATP1B3 Leibovici, 1989
SLC47A1 MATE1 Rapamycin 3.27 Metformin HeLa-MATE1 Meyer, 2010
SLC47A1 MATE1 Rapamycin 3.51 Tetraethylammonium HeLa-MATE1 Meyer, 2010

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Clinical Drug-Drug Interactions

No drug-drug interaction information.


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