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Quercetin

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

No substrate information.


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In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
ABCC4 MRP4 Quercetin 20.8 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
ABCC2 MRP2, cMOAT Quercetin >133 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
ABCC3 MRP3 Quercetin >133 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
SLCO2B1 OATP2B1, OATP-B Quercetin 9.47 Estrone sulfate OATP2B1-expressing oocytes Shirasaka, 2013
ABCC1 MRP1 Quercetin 8.1 Leukotriene C4 MRP1-expressing HeLa vesicles Leslie, 2001
ABCG2 BCRP, MXR Quercetin 0.6 Methotrexate BCRP membrane vesicles Saito, 2006
ABCB11 BSEP Quercetin >133 Taurocholate Sf9 cell membrane vesicles Morgan, 2013

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Clinical Drug-Drug Interactions

No drug-drug interaction information.


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