Transporter |
Synonyms |
Inhibitor |
IC50 (μM) |
Ki (μM) |
Substrate used |
Cell System |
Reference |
SLC22A8 |
OAT3 |
Nitazoxanide |
0.154 |
| 6-CF |
COS-7-OAT3 |
Duan, 2012 |
ABCC2 |
MRP2, cMOAT |
Nitazoxanide |
>133 |
| Estradiol-17beta-glucuronide |
Sf9 cell membrane vesicles |
Morgan, 2013 |
ABCC3 |
MRP3 |
Nitazoxanide |
>133 |
| Estradiol-17beta-glucuronide |
Sf9 cell membrane vesicles |
Morgan, 2013 |
ABCC4 |
MRP4 |
Nitazoxanide |
>133 |
| Estradiol-17beta-glucuronide |
Sf9 cell membrane vesicles |
Morgan, 2013 |
ABCB11 |
BSEP |
Nitazoxanide |
>133 |
| Taurocholate |
Sf9 cell membrane vesicles |
Morgan, 2013 |