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Meloxicam

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

No substrate information.


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In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
SLC22A8 OAT3 Meloxicam 0.54 6-carboxyfluorescein HEK293-OAT3 Zou, 2021
SLC22A6 OAT1 Meloxicam 6.88 6-carboxyfluorescein HEK293-OAT1 Zou, 2021
ABCC3 MRP3 Meloxicam >133 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
ABCC4 MRP4 Meloxicam >133 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
SLCO2B1 OATP2B1, OATP-B Meloxicam 1.59 Estrone sulfate CHO-OATP2B1 Khuri, 2017
ABCB11 BSEP Meloxicam 77.5 Taurocholate Sf9 cell membrane vesicles Morgan, 2013

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Clinical Drug-Drug Interactions

No drug-drug interaction information.


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