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Lesinurad

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

No substrate information.


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In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
SLCO1B1 OATP1B1, OATP-C, OATP2, LST-1 Lesinurad 9.3 Bromsulphthalein MDCK II-OAT1B1 Shen, 2016
SLC22A6 OAT1 Lesinurad 6.99 Urate HEK293-OAT1 Taniguchi, 2019
SLC22A8 OAT3 Lesinurad 1.07 Urate HEK293-OAT3 Taniguchi, 2019

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Clinical Drug-Drug Interactions

No drug-drug interaction information.


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