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Histamine

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Km (μM) Cell System Reference
SLC22A3 OCT3 180 HEK293-OCT3 Grundemann, 1999
SLC22A3 OCT3 220 HEK293-OCT3 Amphoux, 2006
SLC22A2 OCT2 940 HEK293-OCT2 Amphoux, 2006
rat_Slc22a2 OCT2, OCT2r, rOCT2 890 HEK293-rOCT2 Amphoux, 2006
rat_Slc22a3 Oct3 540 HEK293-rOCT3 Amphoux, 2006

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In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
SLC22A3 OCT3 Histamine 140 N-methylpyridinium HEK293-OCT3 Grundemann, 1999

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Clinical Drug-Drug Interactions

No drug-drug interaction information.


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