UCSF home page About UCSF UCSF Medical Center
UCSF home page | About UCSF | UCSF Medical Center

Skip to TransPortal content

Decrease the text sizeRestore original text sizeIncrease the text size Enlarge Text
Click to increase the text size. Restore Text
Click to restore original text size. Reduce Text
Click to decrease the text size.
Transporter Database banner  
Decrease the text size | Restore text size | Increase the text size
 Text Sizer image
Home About and More Information Transporter Data Index
Search:  
 

Glimepiride

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

No substrate information.


Back to top

In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
SLCO1B3 OATP1B3, OATP8 Glimepiride 40.9 Bromsulphthalein HEK293-OATP1B3 Klatt, 2013
SLCO2B1 OATP2B1, OATP-B Glimepiride 1.6 Dibromofluorescein HEK293-OATP2B1 Unger, 2020
SLCO1B1 OATP1B1, OATP-C, OATP2, LST-1 Glimepiride 3.55 Estradiol-17beta-glucuronide HEK-OATP1B1 van, 2013
ABCC3 MRP3 Glimepiride 6.39 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
ABCC4 MRP4 Glimepiride 64 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
SLCO1B1 OATP1B1, OATP-C, OATP2, LST-1 Glimepiride 3.62 Rosuvastatin HEK-OATP1B1 van, 2013
ABCB11 BSEP Glimepiride 15.7 Taurocholate Sf9 cell membrane vesicles Morgan, 2013

Back to top

Clinical Drug-Drug Interactions

No drug-drug interaction information.


Back to top

Contact us | Glossary

Blue banner