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Fenofibrate

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

No substrate information.


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In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
SLCO1B1 OATP1B1, OATP-C, OATP2, LST-1 Fenofibrate 105.2 Estradiol-17beta-glucuronide CHO-OATP1B1 Gui, 2009
ABCC2 MRP2, cMOAT Fenofibrate >133 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
ABCC3 MRP3 Fenofibrate >133 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
ABCC4 MRP4 Fenofibrate >133 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
ABCG2 BCRP, MXR Fenofibrate 170 Rosuvastatin polarized Caco-2 monolayer Elsby, 2016
ABCB11 BSEP Fenofibrate 15.3 Taurocholate Sf9 cell membrane vesicles Morgan, 2013

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Clinical Drug-Drug Interactions

No drug-drug interaction information.


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