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Efonidipine

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

No substrate information.


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In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
ABCB1 MDR1, P-gp Efonidipine 17.3 Daunorubicin MDR1 expressing LLC-PK1 cells Katoh, 2000
ABCB1 MDR1, P-gp Efonidipine 20.6 Daunorubicin MDR1 expressing LLC-PK1 cells Katoh, 2000
ABCB1 MDR1, P-gp Efonidipine 13 Digoxin MDR1 expressing LLC-PK1 cells Takara, 2002

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Clinical Drug-Drug Interactions

No drug-drug interaction information.


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