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Dipyridamole

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

No substrate information.


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In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
SLC22A1 OCT1 Dipyridamole 81 4-(4-dimethylamino)styryl-N-methylpyridinium (ASP+) HEK293-OCT1 Kido, 2011
SLC47A1 MATE1 Dipyridamole 24 4-(4-dimethylamino)styryl-N-methylpyridinium (ASP+) HEK293-MATE1 Kido, 2011
SLC47A1 MATE1 Dipyridamole 26 4-(4-dimethylamino)styryl-N-methylpyridinium (ASP+) HEK293-MATE1 Kido, 2011
SLC47A2 MATE2K Dipyridamole 74 4-(4-dimethylamino)styryl-N-methylpyridinium (ASP+) HEK293-MATE2K Kido, 2011
ABCC4 MRP4 Dipyridamole 2 9-(2-phosphonomethoxyethyl)adenine (PMEA) MRP4-expressing HEK293 vesicles Reid, 2003
ABCC5 MRP5 Dipyridamole 30 9-(2-phosphonomethoxyethyl)adenine (PMEA) MRP4-expressing HEK293 vesicles Reid, 2003
ABCC4 MRP4 Dipyridamole <20 Cholyltaurine MRP4-expressing V79 vesicles Rius, 2003
SLC22A4 OCTN1 Dipyridamole 0.0077 Cytarabine HEK293-hOCTN1 Drenberg, 2017
ABCB1 MDR1, P-gp Dipyridamole 22.7 Daunorubicin NIH-3T3-G185 cells Wang, 2001
SLCO2B1 OATP2B1, OATP-B Dipyridamole 2 Dibromofluorescein HEK293-OATP2B1 Unger, 2020
ABCB1 MDR1, P-gp Dipyridamole 40 Digoxin MDR1 transfected LLC-PK1 Kakumoto, 2002
ABCC4 MRP4 Dipyridamole 8.3 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
ABCC2 MRP2, cMOAT Dipyridamole >133 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
ABCC3 MRP3 Dipyridamole >133 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
ABCB1 MDR1, P-gp Dipyridamole 23.7 LDS-751 NIH-3T3-G185 cells Wang, 2001
ABCB1 MDR1, P-gp Dipyridamole 34.3 Rhodamine 123 NIH-3T3-G185 cells Wang, 2001
ABCB11 BSEP Dipyridamole 4 Taurocholate Sf9 cell membrane vesicles Morgan, 2013

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Clinical Drug-Drug Interactions

No drug-drug interaction information.


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