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Cobicistat

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

No substrate information.


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In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
SLC47A1 MATE1 Cobicistat 4.4 1-methyl-4-phenylpyridinium (MPP+) HEK293-MATE1 Kikuchi, 2019
SLC47A2 MATE2K Cobicistat 3.2 1-methyl-4-phenylpyridinium (MPP+) HEK293-MATE2K Kikuchi, 2019
SLC22A4 OCTN1 Cobicistat 2.49 Tetraethylammonium S2-hOCTN1 DARUNAVIR/COBICISTAT PHARMACOKINETICS WRITTEN SUMMARY

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Clinical Drug-Drug Interactions

No drug-drug interaction information.


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