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Chlorpheniramine

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

No substrate information.


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In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
ABCC2 MRP2, cMOAT Chlorpheniramine >133 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
ABCC3 MRP3 Chlorpheniramine >133 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
ABCC4 MRP4 Chlorpheniramine >133 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
ABCB11 BSEP Chlorpheniramine >133 Taurocholate Sf9 cell membrane vesicles Morgan, 2013
SLC47A1 MATE1 Chlorpheniramine 87.6 Tetraethylammonium HEK293-MATE1 Tsuda, 2009
SLC47A2 MATE2K Chlorpheniramine 191.2 Tetraethylammonium HEK293-MATE2 Tsuda, 2009

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Clinical Drug-Drug Interactions

No drug-drug interaction information.


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