UCSF home page About UCSF UCSF Medical Center
UCSF home page | About UCSF | UCSF Medical Center

Skip to TransPortal content

Decrease the text sizeRestore original text sizeIncrease the text size Enlarge Text
Click to increase the text size. Restore Text
Click to restore original text size. Reduce Text
Click to decrease the text size.
Transporter Database banner  
Decrease the text size | Restore text size | Increase the text size
 Text Sizer image
Home About and More Information Transporter Data Index
Search:  
 

Cerivastatin

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

No substrate information.


Back to top

In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
SLCO1B1 OATP1B1, OATP-C, OATP2, LST-1 Cerivastatin 1.7 Estradiol-17beta-glucuronide HEK-OATP1B1 Hinton, 2008
ABCG2 BCRP, MXR Cerivastatin 18.1 Estrone sulfate BCRP-expressing HEK293 vesicles Hirano, 2005
SLCO2B1 OATP2B1, OATP-B Cerivastatin 66.2 Estrone sulfate MDCK II-OATP2B1 Grube, 2006
SLC22A5 OCTN2 Cerivastatin 425 L-carnitine MDCKII-hOCTN2 Diao, 2009
ABCB11 BSEP Cerivastatin 11.4 Taurocholate BSEP-expressing HEK293 vesicles Hirano, 2005

Back to top

Clinical Drug-Drug Interactions

No drug-drug interaction information.


Back to top

Contact us | Glossary

Blue banner