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Celecoxib

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

No substrate information.


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In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
SLC22A8 OAT3 Celecoxib >200 6-carboxyfluorescein HEK293-OAT3 Zou, 2021
SLC22A6 OAT1 Celecoxib >200 6-carboxyfluorescein HEK293-OAT1 Zou, 2021
SLCO2B1 OATP2B1, OATP-B Celecoxib 13.7 Dibromofluorescein HEK293-OATP2B1 Unger, 2020
ABCC2 MRP2, cMOAT Celecoxib >133 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
ABCC3 MRP3 Celecoxib >133 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
ABCC4 MRP4 Celecoxib >133 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
ABCC4 MRP4 Celecoxib 35 Methotrexate MRP4-expressing HEK293 vesicles El-Sheikh, 2007
ABCB11 BSEP Celecoxib >133 Taurocholate Sf9 cell membrane vesicles Morgan, 2013

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Clinical Drug-Drug Interactions

No drug-drug interaction information.


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