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Home | About and More Information | Transporter Data Index |
Transporter | Synonyms | Km (μM) | Cell System | Reference |
---|---|---|---|---|
SLC22A1 | OCT1 | 23 | HEK293-OCT1 | Chen, 2017 |
SLC47A1 | MATE1 | 28.9 | HEK293-MATE1 | Chen, 2017 |
Transporter | Synonyms | Inhibitor | IC50 (μM) | Ki (μM) | Substrate used | Cell System | Reference |
---|---|---|---|---|---|---|---|
SLC22A1 | OCT1 | Butylscopolamine | 28 | 1-methyl-4-phenylpyridinium (MPP+) | HEK293-OCT1 | Chen, 2017 | |
SLC47A1 | MATE1 | Butylscopolamine | 8.2 | 1-methyl-4-phenylpyridinium (MPP+) | HEK293-MATE1 | Chen, 2017 | |
SLC47A2 | MATE2K | Butylscopolamine | 38.2 | 1-methyl-4-phenylpyridinium (MPP+) | HEK293-MATE2K | Chen, 2017 | |
SLC22A1 | OCT1 | Butylscopolamine | 16 | N-methylpyridinium | HEK293-OCT1 | Muller, 2005 | |
SLC22A2 | OCT2 | Butylscopolamine | 764 | N-methylpyridinium | HEK293-OCT2 | Muller, 2005 |
No drug-drug interaction information.
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