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Bromocriptine

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

No substrate information.


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In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
ABCB1 MDR1, P-gp Bromocriptine 2.81 Calcein AM MDR1-expressing LLC-PK1 cells Ekins, 2002
SLCO1B1 OATP1B1, OATP-C, OATP2, LST-1 Bromocriptine 0.7 Fluorescein-Methotrexate CHO-OATP1B1 Gui, 2010
SLC22A5 OCTN2 Bromocriptine 16.6 L-carnitine MDCKII-hOCTN2 Diao, 2009
ABCB1 MDR1, P-gp Bromocriptine 3.96 Vinblastine MDR1-expressing LLC-PK1 cells Ekins, 2002

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Clinical Drug-Drug Interactions

No drug-drug interaction information.


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