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Home | About and More Information | Transporter Data Index |
No substrate information.
Transporter | Synonyms | Inhibitor | IC50 (μM) | Ki (μM) | Substrate used | Cell System | Reference |
---|---|---|---|---|---|---|---|
SLC22A8 | OAT3 | Bisphenol A | 9.2 | Estrone sulfate | HEK293 cells | Bruyere, 2017 | |
SLCO1B1 | OATP1B1, OATP-C, OATP2, LST-1 | Bisphenol A | 18.7 | Estrone sulfate | CHO cells | Bruyere, 2017 | |
SLC22A1 | OCT1 | Bisphenol A | 39 | Tetraethylammonium | HEK293 cells | Bruyere, 2017 | |
SLC47A1 | MATE1 | Bisphenol A | 73.5 | Tetraethylammonium | HEK293 cells | Bruyere, 2017 |
No drug-drug interaction information.
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