UCSF home page About UCSF UCSF Medical Center
UCSF home page | About UCSF | UCSF Medical Center

Skip to TransPortal content

Decrease the text sizeRestore original text sizeIncrease the text size Enlarge Text
Click to increase the text size. Restore Text
Click to restore original text size. Reduce Text
Click to decrease the text size.
Transporter Database banner  
Decrease the text size | Restore text size | Increase the text size
 Text Sizer image
Home About and More Information Transporter Data Index
Search:  
 

Allethrin

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

No substrate information.


Back to top

In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
SLC22A1 OCT1 Allethrin 2.6 4',6'-diamidino-2-phenylindole HEK293 cells Chedik, 2017
ABCC2 MRP2, cMOAT Allethrin 48.2 Carboxy-2',7'-dichlorofluorescein diacetate HuH-7 cells Chedik, 2017
SLCO1B1 OATP1B1, OATP-C, OATP2, LST-1 Allethrin 16.5 Estrone sulfate CHO cells Chedik, 2017
SLC22A8 OAT3 Allethrin 69.4 Fluorescein HEK293 cells Chedik, 2017
ABCG2 BCRP, MXR Allethrin 42.5 Hoechst 33342 HEK293 cells Chedik, 2017
SLC22A2 OCT2 Allethrin 42.6 Rhodamine 123 HEK293 cells Chedik, 2017
SLC47A1 MATE1 Allethrin 50.2 Tetraethylammonium HEK293 cells Chedik, 2017

Back to top

Clinical Drug-Drug Interactions

No drug-drug interaction information.


Back to top

Contact us | Glossary

Blue banner