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Acetylcholine

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Km (μM) Cell System Reference
SLC22A4 OCTN1 1000 hOCTN1 reconstituted proteoliposome Pochini, 2012

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In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
SLC22A1 OCT1 Acetylcholine 580 1-methyl-4-phenylpyridinium (MPP+) OCT1-expressing oocytes Lips, 2005
SLC22A4 OCTN1 Acetylcholine 440 Tetraethylammonium hOCTN1-reconstituted proteoliposomes Pochini, 2011

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Clinical Drug-Drug Interactions

No drug-drug interaction information.


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