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Acetazolamide

Substrate Information
Inhibitor Information
Clinical Drug-drug Interactions

In Vitro Substrates

No substrate information.


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In Vitro Inhibitors

* denotes drugs that can potentially be used for in vivo (clinical) studies of the designated transporter
Transporter Synonyms Inhibitor IC50 (μM) Ki (μM) Substrate used Cell System Reference
ABCC2 MRP2, cMOAT Acetazolamide >133 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
ABCC3 MRP3 Acetazolamide >133 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
ABCC4 MRP4 Acetazolamide >133 Estradiol-17beta-glucuronide Sf9 cell membrane vesicles Morgan, 2013
SLC22A11 OAT4 Acetazolamide 425 Estrone sulfate S2-OAT4 Hasannejad, 2004
SLC22A8 OAT3 Acetazolamide 816 Estrone sulfate S2-OAT3 Hasannejad, 2004
SLC22A6 OAT1 Acetazolamide 75 Para-aminohippurate S2-OAT1 Hasannejad, 2004
ABCB11 BSEP Acetazolamide >133 Taurocholate Sf9 cell membrane vesicles Morgan, 2013

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Clinical Drug-Drug Interactions

No drug-drug interaction information.


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